Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
AssayType

Assay
Description
Source

Mol
weight
Rot
Bonds
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H acc

LogP

Smiles

DOI

12948 7808 0 None - 1 Human 8.0 pIC50 = 8 Functional
Determined using a cAMP assay in cells overexpressing hGPR61Determined using a cAMP assay in cells overexpressing hGPR61
Guide to Pharmacology 524 12 1 10 2.7 CCOC1=CC(C)=NC(=N1)N(CCOC)S(=O)(=O)C2=CC=C(NCC3=C(F)C=NC=C3F)N=C2OC 37741852
168510218 7808 0 None - 1 Human 8.0 pIC50 = 8 Functional
Determined using a cAMP assay in cells overexpressing hGPR61Determined using a cAMP assay in cells overexpressing hGPR61
Guide to Pharmacology 524 12 1 10 2.7 CCOC1=CC(C)=NC(=N1)N(CCOC)S(=O)(=O)C2=CC=C(NCC3=C(F)C=NC=C3F)N=C2OC 37741852




Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Similar-
ity
Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
Assay
Type
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI