Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
AssayType

Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI

131648253 9814 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
155817507 9814 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
9139 9814 0 None - 1 Mouse 10.7 pEC50 = 10.7 Functional
High affinity binding site of mouse GPR83High affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
131648253 9814 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
155817507 9814 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
9139 9814 0 None - 1 Mouse 7.0 pEC50 = 7.0 Functional
Low affinity binding site of mouse GPR83Low affinity binding site of mouse GPR83
Guide to Pharmacology None None None None 27117253
32051 10923 0 None - 1 Mouse 5.0 pEC50 = 5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 64 0 0 0 -0.0 [Zn+2] 23335960
566 10923 0 None - 1 Mouse 5.0 pEC50 = 5 Functional
UnclassifiedUnclassified
Guide to Pharmacology 64 0 0 0 -0.0 [Zn+2] 23335960




Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Similar-
ity
Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
Assay
Type
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI

9140 9813 0 None - 1 Mouse 8.1 pKd = 8.1 Binding
N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.N-terminally tyrosinated radioidodinated rPEN binding to mouse GPR83 in hypothalamic membrane preparations.
Guide to Pharmacology None None None None 27117253