Ligand source activities (1 row/activity)





Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
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name
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# Tested
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p-value
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11337 9702 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Measuring β-arrestin recruitment using the PathHunter assay system.Measuring β-arrestin recruitment using the PathHunter assay system.
Guide to Pharmacology 440 4 0 4 3.9 O=c1c2CN(CCc2n2c(=NCC2)n1Cc1ccc(cc1)C(F)(F)F)Cc1ccccc1 31127149
124085867 9702 0 None - 1 Human 6.4 pEC50 = 6.4 Functional
Measuring β-arrestin recruitment using the PathHunter assay system.Measuring β-arrestin recruitment using the PathHunter assay system.
Guide to Pharmacology 440 4 0 4 3.9 O=c1c2CN(CCc2n2c(=NCC2)n1Cc1ccc(cc1)C(F)(F)F)Cc1ccccc1 31127149
5312830 6976 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715
5567 6976 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715
CHEMBL1230670 6976 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715
DB07302 6976 0 None - 1 Human 5.7 pEC50 = 5.7 Functional
UnclassifiedUnclassified
Guide to Pharmacology 296 14 2 2 4.9 CCCCC/C=C\C=C\[C@H](CCCCCCCC(=O)O)O 16236715
12945 9644 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 351 6 2 4 4.0 CC1=C(OC2=C1C=C(NC(=O)CCC(=O)C3=CC=CC=C3)C=C2)C(O)=O 37770763
168654812 9644 0 None - 1 Human 7.3 pEC50 = 7.3 Functional
UnclassifiedUnclassified
Guide to Pharmacology 351 6 2 4 4.0 CC1=C(OC2=C1C=C(NC(=O)CCC(=O)C3=CC=CC=C3)C=C2)C(O)=O 37770763
12944 9643 0 None - 1 Human 7.8 pIC50 = 7.8 Functional
Efficacy 90%Efficacy 90%
Guide to Pharmacology 359 6 2 4 3.0 CC1=C(OC2=C1C=C(C=C2)S(=O)(=O)NCCC3=CC=CC=C3)C(O)=O 37770763
4319354 9643 0 None - 1 Human 7.8 pIC50 = 7.8 Functional
Efficacy 90%Efficacy 90%
Guide to Pharmacology 359 6 2 4 3.0 CC1=C(OC2=C1C=C(C=C2)S(=O)(=O)NCCC3=CC=CC=C3)C(O)=O 37770763




Ligands (move mouse cursor over ligand name to see structure) Receptor Assay information Chemical information
Sel. page Similar-
ity
Common
name
GPCRdb
ID
#Vendors

Reference
ligand
Fold
selectivity
# Tested
GPCRs
Species

p-value
(-log)
Activity
Type
Activity
Relation
Activity
Value
Assay
Type
Assay
Description
Source

Mol
weight
Rot
Bonds
H don

H acc

LogP

Smiles

DOI