Ligand source activities (1 row/activity)
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | ||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
AssayType |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
3700 | 10182 | 0 | None | 4 | 2 | Human | 10.1 | pEC50 | = | 10.1 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 | ||||
3697 | 10175 | 0 | None | -2 | 2 | Human | 10.7 | pEC50 | = | 10.7 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 | ||||
3699 | 10179 | 0 | None | -1 | 2 | Human | 10.7 | pEC50 | = | 10.7 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 | ||||
3698 | 10178 | 0 | None | 3 | 2 | Human | 12.5 | pEC50 | = | 12.5 | Functional | Guide to Pharmacology | None | None | None | None | 21693646 |
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Assay information | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Similar- ity |
Common name |
GPCRdb ID |
#Vendors |
Reference ligand |
Fold selectivity |
# Tested GPCRs |
Species |
p-value (-log) |
Activity Type |
Activity Relation |
Activity Value |
Assay Type |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
3699 | 10179 | 0 | None | - | 1 | Human | 8.7 | pKd | = | 8.7 | Binding | Guide to Pharmacology | None | None | None | None | 21909076 |