Ligand source activities (1 row/activity)
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |
|
3699 | 3406 | None | 0 | Human | Functional | pEC50 | = | 11 | 11.0 | 1 | 2 | Guide to Pharmacology | None | None | None | None | 21693646 | |||||
3697 | 3402 | None | 0 | Human | Functional | pEC50 | = | 11.1 | 11.1 | 2 | 2 | Guide to Pharmacology | None | None | None | None | 21693646 | |||||
3698 | 3405 | None | 0 | Human | Functional | pEC50 | = | 12 | 12.0 | -3 | 2 | Guide to Pharmacology | None | None | None | None | 21693646 | |||||
3700 | 3408 | None | 0 | Human | Functional | pEC50 | = | 9.4 | 9.4 | -4 | 2 | Guide to Pharmacology | None | None | None | None | 21693646 |
Ligands (move mouse cursor over ligand name to see structure) | Receptor | Activity | Chemical information | |||||||||||||||||||
---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Sel. page | Common name |
GPCRdb ID |
Reference ligand |
Vendors |
Species |
Assay Type |
Activity Type |
Activity Relation |
Activity Value |
p-value (-log) |
Fold selectivity |
Tested GPCRs |
Assay Description |
Source |
Mol weight |
Rot Bonds |
H don |
H acc |
LogP |
Smiles |
DOI |