MC1 receptor (mshr_eulfu)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC1 receptor

GENE

MC1R

ORGANISM

Brown lemur (Eulemur fulvus fulvus)

ALT. NAMES

Melanocyte-stimulating hormone receptor, MSH-R, Melanocortin receptor 1, MC1-R

SOURCE

SWISSPROT

SEQUENCE

N-term        
M
P
A
Q
G
S
Q
R
G
L
10
                   
L
G
A
V
N
F
T
P
T
A
20
                   
T
P
H
L
R
P
A
A
N
Q
30
                   
T
G
P
Q
C
L
E
V
S
V
40
TM1              
P
D
G
L
F
L
C
L
G
L
50
                   
V
S
L
V
E
N
T
L
V
V
60
            ICL1
A
A
I
A
K
N
R
N
L
H
70
TM2              
S
P
M
Y
C
F
I
C
C
L
80
                   
A
L
S
D
L
L
V
S
V
S
90
                   
N
L
L
E
T
A
V
L
L
L
100
        ECL1    
L
E
V
G
A
L
A
A
Q
A
110
TM3              
T
V
V
Q
Q
L
G
N
V
I
120
                   
D
V
L
I
C
S
S
M
V
S
130
                   
S
L
C
S
L
G
A
I
A
M
140
                   
D
R
Y
I
S
I
F
Y
A
L
150
ICL2     TM4  
R
Y
H
S
I
V
T
L
A
R
160
                   
A
R
R
A
I
A
A
V
W
A
170
                   
A
S
I
L
S
S
T
L
F
I
180
    ECL2 TM5  
T
Y
Y
D
R
T
A
A
L
L
190
                   
C
L
V
V
F
F
L
A
M
L
200
                   
V
L
M
A
L
L
Y
V
H
M
210
                   
L
I
Q
A
C
Q
H
A
Q
A
220
            ICL3
I
A
R
L
H
K
R
Q
H
P
230
    TM6          
V
Q
Q
G
W
G
L
K
G
A
240
                   
A
T
L
T
I
L
L
G
V
F
250
                   
F
L
C
W
G
P
F
F
L
H
260
                   
L
T
L
I
A
V
C
P
Q
H
270
ECL3            
P
T
C
S
C
I
F
K
N
F
280
TM7              
R
L
F
L
A
L
I
I
C
N
290
                   
T
I
V
D
P
L
I
Y
A
F
300
  H8              
R
S
Q
E
L
R
R
T
L
K
310
C-term  
E
V
L
L
F
S
W

LINKS

DIAGRAMS

7TM

ICL1 R N L H ICL1ECL1 A L A A ECL1ICL2 A L R Y H S I V ICL2ECL2 Y D ECL2ICL3 R Q H P V Q ICL3ECL3 P Q H P T C S C I F K ECL3N-term M P A Q G S Q R G L L G A V N F T P T A T P H L R P A A N Q T G P Q C L E V S V N-termC-term L K E V L L F S W C-term P D G L F L C L G L V S L V E N T L V V A A I A K N S P M Y C F I C C L A L S D L L V S V S N L L E T A V L L L L E V G Q A T V V Q Q L G N V I D V L I C S S M V S S L C S L G A I A M D R Y I S I F Y T L A R A R R A I A A V W A A S I L S S T L F I T Y R T A A L L C L V V F F L A M L V L M A L L Y V H M L I Q A C Q H A Q A I A R L H K Q G W G L K G A A T L T I L L G V F F L C W G P F F L H L T L I A V C N F R L F L A L I I C N T I V D P L I Y A F R S Q E L R R T
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

T N E V L S V L G L C L F L G D P 1 C C L A L S D L L V S V S N L L E T A V 2 A G L S C L S S V M S S C I L V D I V N 3 A R R A I A A V W A A S I L S S T L F I 4 Y L L A M L V L M A L F F V V L C L L A 5 T I L L G V F F L C W G P F F L H L T L 6 L P D V I T N C I I L A L F L R F N 7
Pick color:
 
 
 
 
 
 
 
 
 
 
 
 




Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available