MC2 receptor (a0a067zg92_megam)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Chinese blunt snout bream (Megalobrama amblycephala)

ALT. NAMES

Melanocortin receptor 2

SOURCE

TREMBL

SEQUENCE

N-term        
M
N
S
S
T
E
A
P
F
T
10
                   
N
P
T
D
C
A
E
V
K
V
20
TM1              
P
S
Q
V
F
L
A
I
A
V
30
                   
A
S
L
S
E
N
L
L
V
I
40
            ICL1
V
A
V
I
K
N
K
N
L
H
50
TM2              
S
P
M
Y
C
F
I
C
N
L
60
                   
A
L
F
N
T
I
S
S
L
S
70
                   
K
A
L
E
D
V
L
L
L
F
80
        ECL1    
I
D
A
G
H
L
N
S
R
G
90
TM3              
P
F
E
L
K
I
D
D
I
M
100
                   
D
S
L
T
L
M
G
F
L
G
110
                   
S
I
F
S
I
L
A
I
A
V
120
                   
D
R
Y
I
S
I
F
H
A
L
130
ICL2     TM4  
R
Y
H
T
L
M
T
M
R
R
140
                   
V
V
V
I
L
S
A
I
W
V
150
                   
L
C
G
T
S
G
A
L
M
I
160
      ECL2 TM5
G
F
F
V
A
A
T
V
Q
I
170
                   
F
F
V
V
L
F
F
T
A
L
180
                   
L
L
I
L
L
L
Y
V
H
M
190
                   
F
L
L
A
R
H
H
A
N
R
200
    ICL3        
I
A
S
M
P
G
A
Q
A
R
210
        TM6      
H
R
Q
S
G
L
R
G
A
L
220
                   
T
L
T
I
L
I
G
V
F
V
230
                   
A
C
W
A
P
F
L
F
H
L
240
            ECL3
L
I
M
M
I
C
P
E
N
P
250
TM7              
Y
C
E
C
Y
R
S
L
F
Q
260
                   
L
H
V
V
L
L
V
S
H
A
270
                   
V
I
D
P
A
I
Y
A
F
R
280
H8                
S
A
E
L
R
N
T
Y
K
I
290
                   
M
F
L
H
S
A
A
R
I
C
300
C-term
K
Q
C
V

LINKS

DIAGRAMS

7TM

ICL1 K N L H ICL1ECL1 H L N S R ECL1ICL2 A L R Y H T L M ICL2ECL2 V ECL2ICL3 S M P G A Q A R H R Q S ICL3ECL3 P E ECL3N-term M N S S T E A P F T N P T D C A E V K V N-termC-term A A R I C K Q C V C-term P S Q V F L A I A V A S L S E N L L V I V A V I K N S P M Y C F I C N L A L F N T I S S L S K A L E D V L L L F I D A G G P F E L K I D D I M D S L T L M G F L G S I F S I L A I A V D R Y I S I F H T M R R V V V I L S A I W V L C G T S G A L M I G F F A A T V Q I F F V V L F F T A L L L I L L L Y V H M F L L A R H H A N R I A G L R G A L T L T I L I G V F V A C W A P F L F H L L I M M I C N P Y C E C Y R S L F Q L H V V L L V S H A V I D P A I Y A F R S A E Y K I S L R N T M F L H
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E S L S A V A I A L F V Q S P 1 C N L A L F N T I S S L S K A L E D V L 2 A L I S F I S G L F G M L T L S D M I D 3 V V V I L S A I W V L C G T S G A L M I 4 Y L L L I L L L A T F F L V V F F I Q V 5 T I L I G V F V A C W A P F L F H L L I 6 A P D I V A H S V L L V V H L Q F L S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available