MC2 receptor (a0a1u7s1y6_allsi)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Chinese alligator (Alligator sinensis)

ALT. NAMES

Adrenocorticotropic hormone receptor, Adrenocorticotropin receptor, Melanocortin receptor 2

SOURCE

TREMBL

SEQUENCE

N-term        
M
R
T
D
R
A
S
E
I
I
10
                   
R
L
L
G
Q
T
S
I
P
S
20
                   
S
E
N
I
S
A
L
S
L
N
30
                   
R
T
D
C
T
Q
V
V
V
P
40
TM1              
E
E
V
F
F
T
I
A
A
V
50
                   
G
I
L
E
N
L
L
V
L
I
60
          ICL1  
A
V
I
R
N
K
N
L
H
L
70
TM2              
P
M
Y
F
F
I
C
S
L
A
80
                   
V
S
D
M
L
G
S
L
Y
K
90
                   
T
L
E
N
I
L
I
I
L
C
100
      ECL1      
K
M
G
Y
L
K
P
R
G
D
110
TM3              
F
E
T
K
M
D
D
V
I
D
120
                   
S
M
F
I
L
S
L
L
G
S
130
                   
I
F
S
L
L
T
I
A
A
D
140
                   
R
Y
I
T
I
F
Y
A
L
R
150
ICL2   TM4    
Y
H
N
I
M
T
L
K
R
A
160
                   
L
I
I
L
A
A
I
W
T
F
170
                   
C
A
G
S
G
I
A
I
A
I
180
    ECL2 TM5  
F
S
H
E
T
A
V
V
I
S
190
                   
F
T
I
L
F
P
L
M
L
I
200
                   
F
I
L
C
L
Y
I
H
M
F
210
                   
L
L
A
R
S
H
A
K
K
I
220
  ICL3          
A
S
L
P
T
S
T
V
H
Q
230
    TM6          
R
T
N
T
K
G
A
I
T
L
240
                   
T
I
F
L
G
V
F
L
F
C
250
                   
W
A
P
F
V
L
H
I
L
L
260
        ECL3 TM7
M
Q
F
C
P
H
N
P
Y
C
270
                 
A
C
Y
M
S
I
F
Q
V
N
280
                   
G
T
L
I
L
C
N
A
V
I
290
                H8
D
P
M
V
Y
A
F
R
S
P
300
                   
E
L
W
S
T
F
K
K
M
F
310
      C-term
C
C
T
R
S
N
W
K

LINKS

DIAGRAMS

7TM

ICL1 K N L H ICL1ECL1 Y L K P R ECL1ICL2 A L R Y H N I M ICL2ECL2 H ECL2ICL3 S L P T S T V H Q R T ICL3ECL3 P H ECL3N-term M R T D R A S E I I R L L G Q T S I P S S E N I S A L S L N R T D C T Q V V V N-termC-term R S N W K C-term P E E V F F T I A A V G I L E N L L V L I A V I R N L P M Y F F I C S L A V S D M L G S L Y K T L E N I L I I L C K M G G D F E T K M D D V I D S M F I L S L L G S I F S L L T I A A D R Y I T I F Y T L K R A L I I L A A I W T F C A G S G I A I A I F S E T A V V I S F T I L F P L M L I F I L C L Y I H M F L L A R S H A K K I A N T K G A I T L T I F L G V F L F C W A P F V L H I L L M Q F C N P Y C A C Y M S I F Q V N G T L I L C N A V I D P M V Y A F R S P E F K K T L W S T M F C C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E L I G V A A I T F F V E E P 1 C S L A V S D M L G S L Y K T L E N I L 2 T L L S F I S G L L S L I F M S D I V D 3 A L I I L A A I W T F C A G S G I A I A 4 Y L C L I F I L M L P F L I T F S I V V 5 T I F L G V F L F C W A P F V L H I L L 6 M P D I V A N C L I L T G N V Q F I S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available