MC2 receptor (a0a674ix92_terca)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Three-toed box turtle (Terrapene carolina triunguis)

ALT. NAMES

Adrenocorticotropic hormone receptor, Adrenocorticotropin receptor, Melanocortin receptor 2

SOURCE

TREMBL

SEQUENCE

N-term        
M
R
P
D
S
A
S
Q
I
M
10
                   
R
L
L
G
Q
T
R
I
P
S
20
                   
F
E
N
I
S
N
L
S
M
N
30
                   
S
D
C
T
Q
V
V
V
P
E
40
TM1              
E
V
F
F
T
I
A
I
A
G
50
                   
I
L
E
N
L
L
V
L
I
A
60
        ICL1    
V
I
K
N
K
N
L
H
L
P
70
TM2              
M
Y
L
F
I
C
S
L
S
V
80
                   
S
D
M
L
V
S
L
Y
K
T
90
                   
L
E
N
I
L
I
I
L
G
K
100
    ECL1   TM3
M
G
Y
L
T
P
R
G
D
L
110
                   
E
T
K
I
D
D
V
M
D
S
120
                   
L
F
V
L
S
L
L
G
S
V
130
                   
F
S
L
L
A
I
A
A
D
R
140
            ICL2
Y
I
T
I
F
F
A
L
Q
Y
150
        TM4      
H
N
I
M
T
L
N
R
A
L
160
                   
I
I
L
A
V
I
W
A
F
C
170
                   
A
G
S
G
I
A
M
T
I
F
180
  ECL2 TM5    
S
H
E
T
A
T
V
I
S
F
190
                   
T
I
L
F
P
F
M
L
I
F
200
                   
I
L
C
L
Y
I
H
M
F
L
210
                   
L
A
R
T
H
A
K
K
I
A
220
ICL3            
S
L
P
T
S
A
V
P
Q
R
230
  TM6            
V
N
L
K
G
A
I
T
L
T
240
                   
I
F
F
G
V
F
L
C
C
W
250
                   
G
P
F
L
L
H
I
L
L
M
260
      ECL3 TM7
K
F
C
P
L
N
P
Y
C
A
270
                   
C
Y
M
S
I
F
H
V
N
A
280
                   
T
L
I
L
C
N
G
I
I
D
290
              H8  
P
M
I
Y
A
F
R
S
P
E
300
                   
L
R
S
T
L
K
K
M
F
C
310
    C-term    
C
T
R
Q
A
S
F
F
F
K
320
           
V
S
K
M
S
H

LINKS

DIAGRAMS

7TM

ICL1 K N L H ICL1ECL1 Y L T P R ECL1ICL2 A L Q Y H N I M ICL2ECL2 H ECL2ICL3 S L P T S A V P Q R V ICL3ECL3 P L ECL3N-term M R P D S A S Q I M R L L G Q T R I P S F E N I S N L S M N S D C T Q V V V N-termC-term R Q A S F F F K V S K M S H C-term P E E V F F T I A I A G I L E N L L V L I A V I K N L P M Y L F I C S L S V S D M L V S L Y K T L E N I L I I L G K M G G D L E T K I D D V M D S L F V L S L L G S V F S L L A I A A D R Y I T I F F T L N R A L I I L A V I W A F C A G S G I A M T I F S E T A T V I S F T I L F P F M L I F I L C L Y I H M F L L A R T H A K K I A N L K G A I T L T I F F G V F L C C W G P F L L H I L L M K F C N P Y C A C Y M S I F H V N A T L I L C N G I I D P M I Y A F R S P E L K K T L R S T M F C C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E L I G A I A I T F F V E E P 1 C S L S V S D M L V S L Y K T L E N I L 2 A L L S F V S G L L S L V F L S D M V D 3 A L I I L A V I W A F C A G S G I A M T 4 Y L C L I F I L M F P F L I T F S I V T 5 T I F F G V F L C C W G P F L L H I L L 6 M P D I I G N C L I L T A N V H F I S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available