MC2 receptor (a0a6i9xj90_9saur)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Thamnophis sirtalis (Thamnophis sirtalis)

ALT. NAMES

Adrenocorticotropic hormone receptor, Adrenocorticotropin receptor, Melanocortin receptor 2

SOURCE

TREMBL

SEQUENCE

N-term        
M
K
T
N
T
A
S
E
I
I
10
                   
R
L
L
E
Q
R
S
M
H
I
20
                   
F
E
N
Q
S
E
Q
S
L
N
30
                   
V
S
N
C
M
S
I
V
V
P
40
TM1              
E
E
I
F
F
T
I
A
T
V
50
                   
G
I
L
E
N
L
L
V
L
I
60
          ICL1  
A
V
G
R
N
K
N
L
H
S
70
TM2              
P
M
Y
I
F
I
C
S
L
A
80
                   
V
S
D
M
L
G
S
L
S
K
90
                   
T
M
E
N
I
F
Y
I
I
F
100
      ECL1      
C
K
M
K
Y
L
P
C
H
G
110
TM3              
N
M
A
R
T
V
D
D
V
I
120
                   
D
F
M
F
I
L
S
L
L
G
130
                   
S
I
F
S
L
S
V
I
A
A
140
                   
D
R
Y
I
T
I
F
Y
A
L
150
ICL2     TM4  
R
Y
H
N
I
M
T
Q
K
R
160
                   
A
L
L
I
L
L
V
I
W
A
170
                   
F
C
A
G
S
G
I
A
M
V
180
      ECL2 TM5
I
F
S
F
E
T
A
T
V
I
190
                   
S
F
S
A
L
F
S
F
M
L
200
                   
I
F
I
L
C
L
Y
I
H
M
210
                   
F
M
L
G
R
S
H
A
I
K
220
    ICL3        
I
A
L
M
S
A
S
S
V
Q
230
      TM6        
Q
R
I
N
M
K
G
T
I
T
240
                   
L
T
V
L
L
G
V
F
L
C
250
                   
C
W
A
P
F
V
L
H
I
L
260
          ECL3 TM7
L
I
Q
F
C
P
R
N
P
Y
270
               
C
I
C
Y
L
S
I
F
H
V
280
                   
N
G
M
L
I
M
F
N
A
V
290
                   
I
D
P
M
I
Y
A
F
R
S
300
H8                
P
E
L
R
S
T
F
K
R
L
310
        C-term
F
C
C
W
Q
P
S
W
T

LINKS

DIAGRAMS

7TM

ICL1 K N L H ICL1ECL1 K Y L P C H ECL1ICL2 A L R Y H N I M ICL2ECL2 F ECL2ICL3 L M S A S S V Q Q R I ICL3ECL3 P R ECL3N-term M K T N T A S E I I R L L E Q R S M H I F E N Q S E Q S L N V S N C M S I V V N-termC-term Q P S W T C-term P E E I F F T I A T V G I L E N L L V L I A V G R N S P M Y I F I C S L A V S D M L G S L S K T M E N I F Y I I F C K M G N M A R T V D D V I D F M F I L S L L G S I F S L S V I A A D R Y I T I F Y T Q K R A L L I L L V I W A F C A G S G I A M V I F S E T A T V I S F S A L F S F M L I F I L C L Y I H M F M L G R S H A I K I A N M K G T I T L T V L L G V F L C C W A P F V L H I L L I Q F C N P Y C I C Y L S I F H V N G M L I M F N A V I D P M I Y A F R S P E F K R W L R S T L F C C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E L I G V T A I T F F I E E P 1 C S L A V S D M L G S L S K T M E N I F 2 V S L S F I S G L L S L I F M F D I V D 3 A L L I L L V I W A F C A G S G I A M V 4 Y L C L I F I L M F S F L A S F S I V T 5 T V L L G V F L C C W A P F V L H I L L 6 M P D I V A N F M I L M G N V H F I S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available