MC2 receptor (g3nhu6_gasac)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Three-spined stickleback (Gasterosteus aculeatus)

ALT. NAMES

Adrenocorticotropic hormone receptor, Adrenocorticotropin receptor, Melanocortin receptor 2

SOURCE

TREMBL

SEQUENCE

N-term        
M
D
T
A
A
A
N
R
S
D
10
            TM1  
C
P
E
V
R
V
P
V
P
L
20
                   
F
F
T
I
G
V
V
S
L
A
30
                   
E
N
L
L
V
V
V
A
V
I
40
    ICL1 TM2  
R
N
R
N
L
H
S
P
M
Y
50
                   
C
F
I
C
S
L
A
A
F
N
60
                   
T
I
A
S
L
T
K
T
W
E
70
                   
N
L
M
I
V
F
A
N
I
G
80
ECL1   TM3    
L
L
E
K
K
G
P
S
E
T
90
                   
N
V
D
D
V
L
D
S
L
L
100
                   
C
M
S
F
V
G
S
I
V
S
110
                   
F
L
A
I
A
A
D
R
Y
I
120
        ICL2    
S
I
F
H
A
L
R
Y
H
N
130
    TM4          
I
M
T
M
R
R
T
R
A
V
140
                   
L
G
V
I
W
T
L
C
G
V
150
                   
S
A
V
L
M
V
R
F
F
D
160
TM5              
S
N
F
I
M
I
C
F
V
V
170
                   
F
F
V
V
S
L
A
I
I
C
180
                   
F
L
Y
V
Y
M
F
M
L
A
190
                   
R
I
H
A
R
K
I
A
A
L
200
ICL3 TM6      
P
A
S
N
G
M
R
G
A
L
210
                   
T
L
T
I
L
F
G
A
F
V
220
                   
V
C
W
A
P
F
F
L
H
L
230
            ECL3
I
I
I
M
L
C
P
T
N
P
240
TM7              
Y
C
E
C
Y
R
S
L
F
Q
250
                   
L
H
V
V
L
L
M
S
H
A
260
                   
F
I
D
P
A
I
Y
A
F
R
270
H8                
S
V
E
L
R
H
T
F
R
K
280
                   
M
L
L
C
S
D
W
K
R
C
290
C-term
S

LINKS

DIAGRAMS

7TM

ICL1 R N L H ICL1ECL1 L L E K K ECL1ICL2 A L R Y H N I M ICL2ECL2 D ECL2ICL3 A L P A S N ICL3ECL3 P T ECL3N-term M D T A A A N R S D C P E V R V N-termC-term D W K R C S C-term P V P L F F T I G V V S L A E N L L V V V A V I R N S P M Y C F I C S L A A F N T I A S L T K T W E N L M I V F A N I G G P S E T N V D D V L D S L L C M S F V G S I V S F L A I A A D R Y I S I F H T M R R T R A V L G V I W T L C G V S A V L M V R F F S N F I M I C F V V F F V V S L A I I C F L Y V Y M F M L A R I H A R K I A G M R G A L T L T I L F G A F V V C W A P F F L H L I I I M L C N P Y C E C Y R S L F Q L H V V L L M S H A F I D P A I Y A F R S V E F R K S L R H T M L L C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E A L S V V G I T F F L P V P 1 C S L A A F N T I A S L T K T W E N L M 2 A L F S V I S G V F S M C L L S D L V D 3 T R A V L G V I W T L C G V S A V L M V 4 Y L F C I I A L S V V F F V V F C I M I 5 T I L F G A F V V C W A P F F L H L I I 6 A P D I F A H S M L L V V H L Q F L S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available