MC2 receptor (h1zyj6_dicla)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

European seabass (Dicentrarchus labrax)

ALT. NAMES

Melanocortin 2 receptor

SOURCE

TREMBL

SEQUENCE

N-term        
M
N
A
N
P
V
N
Q
S
D
10
            TM1  
C
P
E
V
K
V
P
V
P
L
20
                   
F
L
A
I
G
V
V
S
L
A
30
                   
E
N
L
L
V
V
V
A
I
I
40
    ICL1 TM2  
W
N
R
N
L
H
S
P
M
Y
50
                   
C
F
I
C
S
L
A
A
F
N
60
                   
T
I
A
S
L
S
K
T
W
E
70
                   
T
L
M
I
V
F
A
D
V
G
80
ECL1   TM3    
Q
L
E
K
T
G
S
S
V
M
90
                   
K
L
D
D
V
M
D
S
L
L
100
                   
C
M
S
F
V
G
S
I
F
S
110
                   
F
L
A
I
A
V
D
R
Y
I
120
        ICL2    
T
I
F
H
A
L
R
Y
H
N
130
    TM4          
V
M
T
M
R
R
T
G
A
M
140
                   
L
G
I
I
W
T
T
C
G
V
150
                   
V
A
V
L
M
V
R
F
F
D
160
TM5              
S
K
F
I
M
I
C
F
V
A
170
                   
F
F
I
I
S
L
A
I
I
C
180
                   
S
L
Y
V
Y
M
F
M
L
A
190
                   
R
I
H
A
R
K
I
A
A
L
200
ICL3            
P
T
S
S
G
G
R
S
R
H
210
            TM6  
Q
R
W
R
G
N
S
M
R
G
220
                   
A
L
T
L
T
I
L
F
G
A
230
                   
I
V
V
C
W
A
P
F
F
V
240
                   
H
L
I
I
I
M
V
C
P
M
250
TM7              
N
P
Y
C
E
C
Y
R
S
L
260
                   
F
Q
L
H
V
V
L
L
M
S
270
                   
H
S
V
V
D
P
A
I
Y
A
280
    H8            
F
R
I
A
E
L
R
H
T
F
290
                   
R
K
M
L
L
C
S
Q
W
R
300
C-term
R
C
S

LINKS

DIAGRAMS

7TM

ICL1 R N L H ICL1ECL1 Q L E K T ECL1ICL2 A L R Y H N V M ICL2ECL2 D ECL2ICL3 A L P T S S G G R S R H Q R W R G N ICL3ECL3 P M ECL3N-term M N A N P V N Q S D C P E V K V N-termC-term Q W R R C S C-term P V P L F L A I G V V S L A E N L L V V V A I I W N S P M Y C F I C S L A A F N T I A S L S K T W E T L M I V F A D V G G S S V M K L D D V M D S L L C M S F V G S I F S F L A I A V D R Y I T I F H T M R R T G A M L G I I W T T C G V V A V L M V R F F S K F I M I C F V A F F I I S L A I I C S L Y V Y M F M L A R I H A R K I A S M R G A L T L T I L F G A I V V C W A P F F V H L I I I M V C N P Y C E C Y R S L F Q L H V V L L M S H S V V D P A I Y A F R I A E F R K S L R H T M L L C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E A L S V V G I A L F L P V P 1 C S L A A F N T I A S L S K T W E T L M 2 A L F S F I S G V F S M C L L S D M V D 3 T G A M L G I I W T T C G V V A V L M V 4 Y L S C I I A L S I I F F A V F C I M I 5 T I L F G A I V V C W A P F F V H L I I 6 A P D V V S H S M L L V V H L Q F L S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available