MC2 receptor (i3nfr9_icttr)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Thirteen-lined ground squirrel (Ictidomys tridecemlineatus)

ALT. NAMES

Adrenocorticotropic hormone receptor, Adrenocorticotropin receptor, Melanocortin receptor 2

SOURCE

TREMBL

SEQUENCE

N-term        
K
P
L
I
S
A
H
G
P
A
10
                   
N
D
S
A
R
N
N
S
D
C
20
          TM1    
P
H
V
V
L
P
D
E
V
F
30
                   
F
T
I
S
V
V
G
V
L
E
40
                   
N
L
L
V
L
L
A
V
I
R
50
  ICL1 TM2    
N
K
N
L
Q
S
P
M
Y
L
60
                   
F
I
C
S
L
A
V
S
D
M
70
                   
L
G
S
L
Y
K
I
L
E
N
80
                   
I
L
I
M
F
R
N
T
G
Y
90
ECL1 TM3      
L
E
P
R
G
T
F
E
T
T
100
                   
A
D
D
I
I
D
S
L
F
V
110
                   
L
S
L
L
G
S
I
S
S
L
120
                   
S
V
I
A
A
D
R
Y
L
T
130
      ICL2      
I
F
H
A
L
Q
Y
H
S
I
140
  TM4            
M
T
M
R
R
T
V
I
I
L
150
                   
G
V
V
W
T
F
C
T
G
S
160
                   
G
I
T
M
V
I
F
S
H
H
170
TM5              
V
P
T
V
L
T
F
A
S
L
180
                   
F
P
L
M
L
V
F
I
L
G
190
                   
L
Y
V
H
M
F
L
L
A
R
200
                   
S
H
A
R
K
I
S
R
L
P
210
ICL3 TM6      
R
T
N
M
K
G
A
L
T
L
220
                   
T
I
L
L
G
V
F
I
F
C
230
                   
W
A
P
F
V
L
H
I
L
L
240
        ECL3 TM7
M
T
F
C
P
N
N
P
Y
C
250
                 
A
C
Y
M
S
L
F
Q
V
N
260
                   
G
M
L
I
M
C
N
A
V
I
270
                H8
D
P
L
I
Y
A
F
R
S
P
280
                   
E
L
R
Q
A
F
K
N
M
L
290
      C-term
F
C
S
R
C
Q

LINKS

DIAGRAMS

7TM

ICL1 K N L Q ICL1ECL1 Y L E P R ECL1ICL2 A L Q Y H S I M ICL2ECL2 H ECL2ICL3 R L P R T ICL3ECL3 P N ECL3N-term K P L I S A H G P A N D S A R N N S D C P H V V L N-termC-term R C Q C-term P D E V F F T I S V V G V L E N L L V L L A V I R N S P M Y L F I C S L A V S D M L G S L Y K I L E N I L I M F R N T G G T F E T T A D D I I D S L F V L S L L G S I S S L S V I A A D R Y L T I F H T M R R T V I I L G V V W T F C T G S G I T M V I F S H V P T V L T F A S L F P L M L V F I L G L Y V H M F L L A R S H A R K I S N M K G A L T L T I L L G V F I F C W A P F V L H I L L M T F C N P Y C A C Y M S L F Q V N G M L I M C N A V I D P L I Y A F R S P E F K N S L R Q A M L F C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E L V G V V S I T F F V E D P 1 C S L A V S D M L G S L Y K I L E N I L 2 V S L S S I S G L L S L V F L S D I I D 3 T V I I L G V V W T F C T G S G I T M V 4 Y L G L I F V L M L P F L S A F T L V T 5 T I L L G V F I F C W A P F V L H I L L 6 L P D I V A N C M I L M G N V Q F L S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available