MC2 receptor (k7exi3_pelsi)

FAMILY

Class A (Rhodopsin) Peptide receptors Melanocortin receptors MC2 receptor

GENE

MC2R

ORGANISM

Chinese softshell turtle (Pelodiscus sinensis)

ALT. NAMES

Adrenocorticotropic hormone receptor, Adrenocorticotropin receptor, Melanocortin receptor 2

SOURCE

TREMBL

SEQUENCE

N-term        
S
F
E
N
N
S
N
I
S
M
10
                   
N
S
D
C
T
Q
V
V
V
P
20
TM1              
E
E
V
F
F
T
I
A
A
A
30
                   
G
I
L
E
N
L
L
V
L
I
40
          ICL1  
A
V
I
K
N
K
N
L
H
L
50
TM2              
P
M
Y
F
F
I
C
S
L
S
60
                   
V
S
D
I
L
V
S
L
Y
K
70
                   
T
L
E
N
I
L
I
I
L
C
80
      ECL1      
K
M
G
Y
L
T
P
R
G
Y
90
TM3              
F
E
T
K
I
D
D
V
I
D
100
                   
S
L
F
I
L
S
L
L
G
S
110
                   
I
F
S
L
L
A
I
A
A
D
120
                   
R
Y
I
T
I
F
F
A
L
Q
130
ICL2   TM4    
Y
H
N
I
M
T
L
N
R
A
140
                   
L
I
I
L
A
V
I
W
V
V
150
                   
C
A
G
S
G
I
A
I
T
I
160
    ECL2 TM5  
F
S
H
E
T
A
T
V
I
S
170
                   
F
T
I
L
F
P
F
M
L
T
180
                   
F
I
L
C
L
Y
I
H
M
F
190
                   
L
L
A
R
S
H
A
K
K
I
200
  ICL3          
A
S
L
P
T
S
A
V
P
S
210
    TM6          
R
V
N
L
K
G
A
I
T
L
220
                   
T
I
F
L
G
V
F
L
C
C
230
                   
W
G
P
F
L
L
H
I
L
L
240
        ECL3 TM7
V
T
F
C
P
F
N
P
Y
C
250
                 
A
C
Y
M
S
I
F
H
V
N
260
                   
A
T
L
I
L
C
N
G
I
I
270
                H8
D
P
M
I
Y
A
F
R
S
P
280
                   
E
L
R
S
T
L
K
K
M
F
290
      C-term
C
C
T
R
S
D
W

LINKS

DIAGRAMS

7TM

ICL1 K N L H ICL1ECL1 Y L T P R ECL1ICL2 A L Q Y H N I M ICL2ECL2 H ECL2ICL3 S L P T S A V P S R V ICL3ECL3 P F ECL3N-term S F E N N S N I S M N S D C T Q V V V N-termC-term R S D W C-term P E E V F F T I A A A G I L E N L L V L I A V I K N L P M Y F F I C S L S V S D I L V S L Y K T L E N I L I I L C K M G G Y F E T K I D D V I D S L F I L S L L G S I F S L L A I A A D R Y I T I F F T L N R A L I I L A V I W V V C A G S G I A I T I F S E T A T V I S F T I L F P F M L T F I L C L Y I H M F L L A R S H A K K I A N L K G A I T L T I F L G V F L C C W G P F L L H I L L V T F C N P Y C A C Y M S I F H V N A T L I L C N G I I D P M I Y A F R S P E L K K T L R S T M F C C
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

L N E L I G A A A I T F F V E E P 1 C S L S V S D I L V S L Y K T L E N I L 2 A L L S F I S G L L S L I F L S D I V D 3 A L I I L A V I W V V C A G S G I A I T 4 Y L C L I F T L M F P F L I T F S I V T 5 T I F L G V F L C C W G P F L L H I L L 6 M P D I I G N C L I L T A N V H F I S 7
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Invitro Mutant Data: Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A

PHYSIOLOGICAL LIGANDS

No physiological ligands available

STRUCTURE MODELS

No structure models available. Check the Archive on Structure models for earlier releases.

STRUCTURES

No structures available