Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
cnr1_rat 5.67x67 304 TM5 S => A N/A N/A Garcia DE et al (1998)
cnr1_rat 317 ICL3 S => A N/A N/A Garcia DE et al (1998)
cnr1_rat 323 ICL3 S => A N/A N/A Garcia DE et al (1998)
cnr1_rat 317 ICL3 S => A N/A N/A Garcia DE et al (1998)
cnr1_rat 419 C-term T => A N/A N/A Jin W et al (1999)
cnr1_rat 426 C-term S => A N/A N/A Jin W et al (1999)
cnr1_rat 430 C-term S => A N/A N/A Jin W et al (1999)
cnr1_rat 2.50x50 164 TM2 D => N N/A N/A Befort K et al (1999)
cnr1_rat 2.50x50 164 TM2 D => N N/A N/A Roche JP et al (1999)
cnr1_rat 5.67x67 304 TM5 S => A N/A N/A Garcia DE et al (1998)
cnr1_rat 317 ICL3 S => A N/A N/A Garcia DE et al (1998)
cnr1_rat 323 ICL3 S => A N/A N/A Garcia DE et al (1998)
cnr1_rat 7.49x49 394 TM7 N => D N/A N/A Roche JP et al (1999)
cnr1_rat 419 C-term T => A N/A N/A Jin W et al (1999)
cnr1_rat 426 C-term S => A N/A N/A Jin W et al (1999)
cnr1_rat 430 C-term S => A N/A N/A Jin W et al (1999)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 R S L R C ICL1ECL1 F H R K D ECL1ICL2 P L A Y K R I V ICL2ECL2 W N C K K L Q S V C S D I F P L I ECL2ICL3 T Q K S I I I H T S E D G K V Q V T R ICL3ECL3 K M ECL3N-term M K S I L D G L A D T T F R T I T T D L L Y V G S N D I Q Y E D I K G D M A S K L G Y F P Q K F P L T S F R G S P F Q E K M T A G D N S P L V P A G D T T N I T E F Y N K S L S S F K E N E E N I Q C G E N F M D M E C F M I L N-termC-term S C E G T A Q P L D N S M G D S D C L H K H A N N T A S M H R A A E S C I K S T V K I A K V T M S V S T D T S A E A L C-term N P S Q Q L A I A V L S L T L G T F T V L E N L L V L C V I L H S R P S Y H F I G S L A V A D L L G S V I F V Y S F V D F H V S P N V F L F K L G G V T A S F T A S V G S L F L T A I D R Y I S I H R T R P K A V V A F C L M W T I A I V I A V L P L L G D E T Y L M F W I G V T S V L L L F I V Y A Y M Y I L W K A H S H A V R M I Q R G P D Q A R M D I R L A K T L V L I L V V L I I C W G P L L A I M V Y D V F G N K L I K T V F A F C S M L C L L N S T V N P I I Y A L R S K D F R S L R H A M F P
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
L N E L V T F T G L T L S L V A I A L Q 1 G S L A V A D L L G S V I F V Y S F V D 2 L F L S G V S A T F S A T V G G L K F L 3 A V V A F C L M W T I A I V I A V L P L 4 Y A Y V I F L L L V S T V G I W F M L Y 5 V L I L V V L I I C W G P L L A I M V Y 6 I P N V T S N L L C L M S C F A F V T 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
CB1 receptor
TM2
2x50 2.50x50 D164
TM5
5x67 5.67x67 S304
TM7
7x49 7.49x49 N394