Mutant Browser

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Protein name Generic number Position Segment Mutation FoldChange or Qual Exp Type Ligand Reference Review
hrh2_rat 34.51x51 124 ICL2 L => A N/A N/A Smit MJ et al (1996)
hrh2_rat 3.49x49 115 TM3 D => N N/A N/A Alewijnse AE et al (2000)
hrh2_rat 3.49x49 115 TM3 D => A N/A N/A Alewijnse AE et al (2000)
hrh2_rat 3.50x50 116 TM3 R => N N/A N/A Alewijnse AE et al (2000)
hrh2_rat 3.50x50 116 TM3 R => A N/A N/A Alewijnse AE et al (2000)
hrh2_rat 3.49x49 115 TM3 D => A N/A N/A Alewijnse AE et al (2000)
hrh2_rat 3.49x49 115 TM3 D => N N/A N/A Alewijnse AE et al (2000)
hrh2_rat 3.49x49 115 TM3 D => N N/A N/A Hoffmann M et al (2001)
hrh2_rat 3.50x50 116 TM3 R => A N/A N/A Alewijnse AE et al (2000)
hrh2_rat 3.50x50 116 TM3 R => N N/A N/A Alewijnse AE et al (2000)
Protein name Generic number Segment Position Mutation FoldChange or Qual Exp Type Ligand Reference Review


Residue

Diagrams

ICL1 R R L R ICL1ECL1 T W S F ECL1ICL2 P L R Y P V L V ICL2ECL2 W N S R N G T R G G N D T F K C K V Q V ECL2ICL3 H I S ICL3ECL3 G D D A I ECL3N-term M E P N G T V H S N-termC-term C K F A S H N S H K T S L R L N N S L L P R S Q S R E G R W Q E E K P L K L Q V W S G T E L T H P Q G N P I R C-term C C L D S M A L K V T I S V V L T T L I L I T I A G N V V V C L A V S L N S L T N C F I V S L A A T D L L L G L L V L P F S A I Y Q L S F G H V F C N I Y T S L D V M L C T A S I L N L F M I S L D R Y C A V T D T P V R V A I S L V F I W V I S I T L S F L S I H L G N E V Y G L V D G L V T F Y L P L L I M C V T Y Y R I F K I A R E Q A K R I N S W K A A T I R E H K A T V T L A A V M G A F I I C W F P Y F T A F V Y R G L R N E A V E G I V L W L G Y A N S A L N P I L Y A A L N R D Y Q Q F R T A L F H
Download: PNG | SVG Increased binding/potency: >5-fold, >10-fold; Reduced binding/potency: >5-fold, >10-fold; No/low effect (<5-fold); and N/A
V N G A I T I L I L T T L V V S I T V K 1 V S L A A T D L L L G L L V L P F S A I Y 2 M F L N L I S A T C L M V D L S T Y I N 3 V A I S L V F I W V I S I T L S F L S I 4 Y T V C M I L L P L Y F T V L G D V L G Y 5 A A V M G A F I I C W F P Y F T A F V Y 6 I P N L A S N A Y G L W L V I G E V A 7
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Residue Table


GPCRdb(A)
GPCRdb(A)
H2 receptor
TM3
3x49 3.49x49 D115
3x50 3.50x50 R116